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1. L-type calcium channel (CaV1.2)
Channel
Cav1.2/β2/α2/δ1, L-type
Catalog Ref.
ICE-CHO-Cav1.2
Gene
CACNA1C
Sources
human
Expression system
CHO
Method
whole cell patch clamp
Reference Inhibitor
Nifedipine(31.3nM±6.8nM), verapamil
Target
Timothy syndrome, long QT syndrome, Pain, epilepsy, hypertension, stroke, arrhythmia, Autism
2、N-type calcium channel (CaV2.2)
Cav2.2/β3/α2δ1 , N-type
ICE-CHO-Cav2.2
CACNA1B
Reference compound
Nifedipine, verapamil, Cadmium (IC50=7.0µm±704nM)
Pain, Spinal cord injury, Kleefstra syndrome
3、T-type calcium channel (CaV3.2)
CaV3.2, T-type
ICE-CHO-Cav3.2
CACNA1H
HEK293
Nifedipine, verapamil, NiCl
Convulsion
4、P/Q-type calcium channel (CaV2.1)
Cav2.1
ICE-CHO-Cav2.1
CACNA1A
Reference inhibitor
Cadmium (2.9 ± 0.658µM)
migraine, seizure and ataxia syndromes
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